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Collezione AO Ordine Mauriziano

  

Items : 5

Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2-Hydroxypyrazolo[1,5-a]pyridine Scaffold: SAR of the Aryloxyaryl Moiety. in Journal of medicinal chemistry / J Med Chem. 2022 Oct 13;65(19):12701-12724. doi: 10.1021/acs.jmedchem.2c00496. Epub 2022 Sep 26.
2022
AO Ordine Mauriziano

Sainas S; Giorgis M; Circosta P; Poli G; Alberti M; Passoni A; Gaidano V; Pippione AC; Vitale N; Bonanni D; Rolando B; Cignetti A; Ramondetti C; Lanno A; Ferraris DM; Canepa B; Buccinnà B; Piccinini M; Rizzi M; Saglio G; Al-Karadaghi S; Boschi D; Miggiano R; Tuccinardi T; Lolli ML;

Dihydroorotate dehydrogenase inhibition reveals metabolic vulnerability in chronic myeloid leukemia. in Cell death & disease / Cell Death Dis. 2022 Jun 30;13(6):576. doi: 10.1038/s41419-022-05028-9.
2022
AOU Alessandria
AO Ordine Mauriziano

Oliviero S; Taverna D; Castagnetti F; Caocci G; Mulas O; Breccia M; Abruzzese E; Iurlo A; Sora F; Geuna M; Gai M; Passoni A; Fava C; Boschi D; Giorgis M; Gaidano V; Sainas S; Molineris I; Cignetti A; Orso F; Vitale N; Houshmand M; Pane F; Lolli ML; Circosta P; Saglio G;

Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2-Hydroxypyrazolo[1,5-a]pyridine Scaffold: SAR of the Biphenyl Moiety. in Journal of medicinal chemistry / J Med Chem. 2021 May 13;64(9):5404-5428. doi: 10.1021/acs.jmedchem.0c01549. Epub 2021 Apr 12.
2021
AOU Alessandria
AO Ordine Mauriziano

Lolli ML; Saglio G; Boschi D; Al-Karadaghi S; Giraudo E; Cignetti A; Piccinini M; Houshmand M; Buccinnà B; Mishina M; Ramondetti C; Bona A; Rolando B; Canepa B; Cojocaru CF; Qiu Y; Passoni A; Bagnati R; Pippione AC; Bonanni D; Gaidano V; Circosta P; Giorgis M; Sainas S;

The Synergism between DHODH Inhibitors and Dipyridamole Leads to Metabolic Lethality in Acute Myeloid Leukemia. in Cancers / Cancers (Basel). 2021 Feb 28;13(5):1003. doi: 10.3390/cancers13051003.
2021
AOU Alessandria
AO Ordine Mauriziano

Cignetti A; Cilloni D; Lolli ML; Boschi D; Giorgis M; Pippione AC; Sainas S; Rapelli S; Tenace V; Morotti A; Carrà G; Vitale N; Houshmand M; Gaidano V; Saglio G; Circosta P;

Targeting Myeloid Differentiation Using Potent 2-Hydroxypyrazolo[1,5- a]pyridine Scaffold-Based Human Dihydroorotate Dehydrogenase Inhibitors. in Journal of medicinal chemistry / J Med Chem. 2018 Jul 26;61(14):6034-6055. doi: 10.1021/acs.jmedchem.8b00373. Epub 2018 Jul 9.
2018
AO Ordine Mauriziano

Sainas S; Pippione AC; Lupino E; Giorgis M; Circosta P; Gaidano V; Goyal P; Bonanni D; Rolando B; Cignetti A; Ducime A; Andersson M; Järvå M; Friemann R; Piccinini M; Ramondetti C; Buccinnà B; Al-Karadaghi S; Boschi D; Saglio G; Lolli ML;