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Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2-Hydroxypyrazolo[1,5-a]pyridine Scaffold: SAR of the Biphenyl Moiety. in Journal of medicinal chemistry / J Med Chem. 2021 May 13;64(9):5404-5428. doi: 10.1021/acs.jmedchem.0c01549. Epub 2021 Apr 12.
2021
AOU Alessandria
AO Ordine Mauriziano
AOU Alessandria
AO Ordine Mauriziano
Lolli ML; Saglio G; Boschi D; Al-Karadaghi S; Giraudo E; Cignetti A; Piccinini M; Houshmand M; Buccinnà B; Mishina M; Ramondetti C; Bona A; Rolando B; Canepa B; Cojocaru CF; Qiu Y; Passoni A; Bagnati R; Pippione AC; Bonanni D; Gaidano V; Circosta P; Giorgis M; Sainas S;
The Synergism between DHODH Inhibitors and Dipyridamole Leads to Metabolic Lethality in Acute Myeloid Leukemia. in Cancers / Cancers (Basel). 2021 Feb 28;13(5):1003. doi: 10.3390/cancers13051003.
2021
AOU Alessandria
AO Ordine Mauriziano
AOU Alessandria
AO Ordine Mauriziano
Cignetti A; Cilloni D; Lolli ML; Boschi D; Giorgis M; Pippione AC; Sainas S; Rapelli S; Tenace V; Morotti A; Carrà G; Vitale N; Houshmand M; Gaidano V; Saglio G; Circosta P;